Fenobam
Potent and selective non-competitive mGluR5 antagonist that displays inverse agonist properties; blocks mGluR5 constitutive activity in vitro (IC50=87nM). Acts at an allosteric modulatory site shared with MPEP (Prod. No. ALX-550-368) and binds mGluR5 with Kd values of 54nM and 31nM for rat and human receptors respectively. Displays anxiolytic activity following oral administration in vivo.
Product Details
| Category |
API's & Drug Standards |
|---|---|
| Price | POA |
| CAS Number | 57653-26-6 |
| Formula | C11H11ClN4O2 |
| Molecular Weight | 266.68 |
| Purity | 98.0% |
| Appearance | Off-white to pale orange solid. |
| Availability | In Stock |
| Storage Conditions | +4°C |
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