Bestatin Hydrochloride
A metalloprotease inhibitor selective for aminopeptidase. Bestatin is a competitive and specific inhibitor of leucine aminopeptidase, aminopeptidase B, and triamino peptidase. It inhibits aminopeptidase B at 60 nM (using arginine-β-naphthylamide as substrate) and leucine aminopeptidase at 20 nM (leucine-β-naphthylamide as substrate). It showed no inhibition of aminopeptidase A, trypsin, chymotrypsin, elastase, papain, pepsin, or themolysin. It offers promise as a novel analgesic because it protects endogenous opioid peptides against degradation.
Product Details
Category |
Antibiotics & Antibacterials Biochemicals & Diagnostics |
---|---|
Price | Custom packed. Request price on line. |
CAS Number | 65391-42-6 |
Formula | C16H24N2O4 · HCl |
Molecular Weight | 344.87 |
Purity | Min 98% (on anhydrous basis) |
Appearance | White to off white powder |
Availability | In Stock |
Storage Conditions | -18°C |
MDL Number | MFCD00058004 |
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